基本信息
马小锋  男    中国科学院成都生物研究所
电子邮件: maxf@cib.ac.cn
通信地址: 成都市高新区科园南路93号,中国科学院成都生物研究所
邮政编码: 610041

研究领域

有机化学、药物化学

招生信息

   
招生专业
070303-有机化学
100701-药物化学
招生方向
糖化学
不对称催化
有机合成、药物合成

教育背景

2007-09--2012-07   中国科学院成都生物研究所天然产物研究中心   理学博士
2003-09--2007-07   兰州大学 药学院   医学学士

工作经历

2019-09~现在, 中国科学院成都生物研究所天然产物研究中心, 研究员
2016-03~2019-03,英国布里斯托大学化学系, 博士后
2012-12~2016-03,比利时天主教鲁汶大学化学与药物化学系, 博士后
2012-07~2012-10,中国科学院成都生物研究所天然产物研究中心, 研究助理


工作简历
2019-09~现在, 中国科学院成都生物研究所天然产物研究中心, 研究员
2016-03~2019-03,英国布里斯托大学化学系, 博士后
2012-12~2016-03,比利时天主教鲁汶大学化学与药物化学系, 博士后
2012-07~2012-10,中国科学院成都生物研究所天然产物研究中心, 研究助理

专利与奖励

   
专利成果
( 1 ) 一种二苯并[c,e][1,2]氧硫杂环己烷-6-氧化物类化合物的转化方法, 发明, 2019, 第 1 作者, 专利号: 201910893751.3

出版信息

   
发表论文
(1) Post-functionalization of dibenzothiophene to functionalized biphenyls via a photoinduced thia-Baeyer-Villiger oxidation, Nature Communications,2020, doi.org/10.1038/s41467-020-14522-7, 2020-02, 通讯作者
(2) An Effective Method for the Synthesis of 1,3‐Dihydro‐2H‐indazoles via N‐N Bond Formation, Adv. Synth. Catal. 2019, 361, 5552-5557, 2019-12, 第 4 作者
(3) Enantioselective Aza-Heck Cyclizations of N (Tosyloxy)carbamates: Synthesis of Pyrrolidines and Piperidines, J. Am. Chem. Soc. 2019, 141, 3356-3360., 2019-02, 第 1 作者
(4) Synthesis of Diketones, Ketoesters and Tetraketones by Electrochemical Oxidative Decarboxylation of Malonic Acid Derivatives: Application to the Synthesis of cis-Jasmone, J. Org. Chem. 2018, 83, 12044-12055., 2018-09, 第 1 作者
(5) Electrochemical Methoxymethylation of Alcohols–A New, Green and Safe Approach for the Preparation of MOM Ethers and Other Acetals, Chem. Commun. 2018, 54, 9969-9972., 2018-08, 第 2 作者
(6) Oxadiazepine Synthesis by Formal [4+3] Cycloaddition of o‐Chloromethyl Arylsulfonamides with Nitrones Promoted by NaHCO3, Adv. Synth. Catal. 2018, 360, 3015-30189., 2018-08, 第 5 作者
(7) A facile Method for the Synthesis of Fused Perhydropyrano[2,3-b]pyrans Promoted by Yb(OTf)3, Chem. Commun. 2018, 54, 3763-3766., 2018-03, 第 3 作者
(8) A Simple and Broadly Applicable C-N Bond Forming Dearomatization Protocol Enabled by Bifunctional Amino-Reagents, Angew. Chem. Int. Ed. 2017, 56, 14531-14535., 2017-11, 第 1 作者
(9) Transition Metal Free C−N Bond Forming Dearomatizations and Aryl C−H Aminations by in Situ Release of a Hydroxylamine-Based Aminating Agent, J. Am. Chem. Soc. 2017, 139, 14005-14008., 2017-10, 第 2 作者
(10) Diverse N-Heterocyclic Ring Systems via Aza-Heck Cyclizations of N-(Pentafluorobenzoyloxy) sulfonamides, Angew. Chem. Int. Ed. 2016, 55, 11198-11202., 2016-07, 其他(合作组作者)
(11) Straightforward and Effective Synthesis of γ-Aminobutyric Acid Transporter Subtype 2-Selective Acyl-Substituted Azaspiro[4.5]decanes, Bioorg. Med. Chem. Lett. 2016, 26, 417-423., 2015-12, 第 1 作者
(12) Electrochemical Oxidative Decarboxylation of Malonic Acid Derivatives: A Method for the Synthesis of Ketals and Ketones, Org. Lett. 2015, 17, 4690-4693., 2015-09, 第 1 作者
(13) Zn(OTf)2 Promoted Rearrangement of 1,2-Cyclopropanated Sugars with Amines: A Convenient Method for the Synthesis of 3-Polyhydroxyalkyl-substituted Pyrrole Derivatives, Org. Biomol. Chem., 2015, 13, 10865-10873., 2015-09, 第 2 作者
(14) A Neighboring Group Participation Strategy: Direct and Highly Diastereoselective Synthesis of 2-Substituted and 2,2-Bisubstituted Perhydrofuro[2,3-b]pyran Derivatives, Org. Biomol. Chem. 2014, 12, 7381-7388., 2014-07, 第 1 作者
(15) Methanesulfonic Acid-Catalyzed Ring Opening and Glycosylation of 1,2-Cyclopropaneacetylated D-Lyxofuranose, Eur. J. Org. Chem. 2014, 4592- 4599., 2014-07, 第 2 作者
(16) An Efficient and Simple Method for Stereoselective Synthesis of N-substituted Iminosugars from D-Xylose Derivative, Chin. J. Chem. 2014, 32, 361-364, 2014-04, 第 3 作者
(17) Stereospecific [3+2] Cycloaddition of 1,2-Cyclopropanated Sugars and Ketones Catalyzed by SnCl4: an Efficient Synthesis of Multi-Substituted Perhydrofuro[2,3-b]furans and Perhydrofuro[2,3-b]pyrans, Chem. Commun. 2014, 50, 3505-3508., 2014-02, 第 1 作者
(18) InCl3 Catalyzed Highly Diastereoselective [3+2] Cycloaddition of 1,2-Cyclopropanated Sugars with Aldehydes: a Straightforward Synthesis of Persubstituted Bis-Tetrahydrofurans and perhydrofuro [2,3-b]pyrans, Org. Lett. 2013, 15, 5170-5173., 2013-10, 第 1 作者
(19) Straightforward and Highly Diastereoselective Synthesis of 2,2-Disubstituted Perhydrofuro[2,3-b]-pyran (and furan) Derivatives Promoted by BiCl3, Chem. Commun. 2013, 49, 7085-7087, 2013-06, 第 1 作者
(20) A Convenient and Highly Stereoselective Method for Synthesis of Octahydropyrano[3,2-b]pyrrole Derivatives, Carbohydr. Res. 2013, 366, 55-62., 2012-11, 第 1 作者
(21) Stereoselective Synthesis of 2-C-Branched (Acetylmethyl) Oligosaccharides and Glycoconjugates: Lewis Acid-Catalyzed Glycosylation from 1,2-Cyclopropaneacetylated Sugars, J. Org. Chem. 2011, 76, 1045-1053., 2011-12, 第 3 作者
(22) A Practical High-throughput Screening System for Feruloyl Esterases: Substrate Design and Evaluation, J. Mol. Catal.B-Enzym. 2012, 74, 36-40, 2011-09, 其他(合作组作者)
(23) Stereoselective Synthesis of a Series of New N-Alkyl-3-Hydroxypiperidine Derivatives Containing a Hemiketal, Eur. J. Org. Chem. 2011, 4834-4840., 2011-09, 第 3 作者
(24) A Novel and Highly Stereoselective Synthesis of 2-Substituted Perhydrofuro[2,3-b]pyran Derivatives, Org. Lett. 2011, 13, 4276-4279., 2011-07, 第 1 作者
(25) Stereoselective Synthesis of 2-C-Acetonyl-2-Deoxy-D-Galactosides Using 1, 2-Cyclopropanacetylated Sugar as Novel Glycosyl Donor, Org. Lett. 2010, 12, 540-543., 2010-02, 第 3 作者
(26) A Simple and Convenient Method for the Synthesis of Pyranoid Glycals, Carbohydr. Res. 2010, 345, 168-171., 2010-01, 第 3 作者
(27) A Mild and Environmentally Benign Method for the Synthesis of Glycals in PEG-600/H2O, Green Chem. 2009, 11, 1124-1127., 2009-05, 第 3 作者

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